Basket | The Czech Academy of Sciences

1.

0444646 - ÚOCHB 2016 RIV US eng J - Journal Article
Jansa, Petr - Holý, Antonín - Dračínský, Martin - Kolman, Viktor - Janeba, Zlatko - Kmoníčková, Eva - Zídek, Zdeněk
Synthesis and structure-activity relationship studies of polysubstituted pyrimidines as inhibitors of immune-activated nitric oxide production.
Medicinal Chemistry Research. Roč. 24, č. 5 (2015), s. 2154-2166. ISSN 1054-2523. E-ISSN 1554-8120
R&D Projects: GA ČR(CZ) GAP303/12/0172; GA MV VG20102015046
Institutional support: RVO:61388963 ; RVO:68378041
Keywords : pyrimidine * nitric oxide * NO * anti-inflammatory
Subject RIV: CC - Organic Chemistry
Impact factor: 1.436, year: 2015
Permanent Link: http://hdl.handle.net/11104/0247170

2.

0446744 - ÚOCHB 2016 RIV DE eng J - Journal Article
Česnek, Michal - Jansa, Petr - Šmídková, Markéta - Mertlíková-Kaiserová, Helena - Dračínský, Martin - Brust, T. F. - Pávek, P. - Trejtnar, F. - Watts, V. J. - Janeba, Zlatko
Bisamidate Prodrugs of 2-Substituted 9-[2-(Phosphonomethoxy)ethyl]adenine (PMEA, adefovir) as Selective Inhibitors of Adenylate Cyclase Toxin from Bordetella pertussis.
ChemMedChem. Roč. 10, č. 8 (2015), s. 1351-1364. ISSN 1860-7179. E-ISSN 1860-7187
R&D Projects: GA MV VG20102015046
Institutional support: RVO:61388963
Keywords : adenylate cyclase toxin * bisamidates * Bordetella pertussis * nucleosides * phosphonates
Subject RIV: CC - Organic Chemistry
Impact factor: 2.980, year: 2015
Permanent Link: http://hdl.handle.net/11104/0248752

3.

0459500 - ÚEM 2017 RIV NL eng J - Journal Article
Zídek, Zdeněk - Kverka, Miloslav - Dusilová, Adéla - Kmoníčková, Eva - Jansa, Petr
Dual inhibition of nitric oxide and prostaglandin E2 production by polysubstituted 2-aminopyrimidines.
Nitric Oxide-Biology and Chemistry. Roč. 57, jul (2016), s. 48-56. ISSN 1089-8603. E-ISSN 1089-8611
R&D Projects: GA ČR(CZ) GAP303/12/0172
Institutional support: RVO:68378041 ; RVO:61388963
Keywords : pyrimidines * nitric oxide * prostaglandin E-2
Subject RIV: FR - Pharmacology ; Medidal Chemistry; CC - Organic Chemistry (UOCHB-X)
Impact factor: 4.181, year: 2016
Permanent Link: http://hdl.handle.net/11104/0259692

4.

0460505 - BC 2017 RIV NL eng J - Journal Article
Špak, Josef - Janeba, Zlatko - Jansa, Petr - Baszczyňski, Ondřej - Pavingerová, Daniela - Špaková, Vlastimila
Phytotoxicity of acyclic nucleoside phosphonates in Brassica pekinensis and Solanum lycopersicum.
Plant Cell, Tissue and Organ Culture. Roč. 125, č. 2 (2016), s. 375-379. ISSN 0167-6857. E-ISSN 1573-5044
Institutional support: RVO:60077344 ; RVO:61388963
Keywords : Chemotherapy * Virus eradication * Phytotoxicity
Subject RIV: EE - Microbiology, Virology; CC - Organic Chemistry (UOCHB-X)
Impact factor: 2.002, year: 2016
Permanent Link: http://hdl.handle.net/11104/0260564

5.

0470846 - ÚOCHB 2017 RIV NL eng J - Journal Article
Jansa, Petr - Čechová, Lucie - Janeba, Zlatko
A complete degradation of organophosphates by microwave-assisted hydrolysis.
Current Microwave Chemistry. Roč. 3, č. 3 (2016), s. 219-226. ISSN 2213-3356
R&D Projects: GA MV VG20102015046
Institutional support: RVO:61388963
Keywords : organophosphates * microwave irradiation * hydrolysis
OECD category: Organic chemistry
Permanent Link: http://hdl.handle.net/11104/0268383

6.

0471547 - ÚOCHB 2017 RIV GB eng J - Journal Article
Elbert, Tomáš - Hezký, Petr - Jansa, Petr
Synthesis of the derivatives of 6-amino-uracil labelled with C-14.
Journal of Labelled Compounds and Radiopharmaceuticals. Roč. 59, č. 14 (2016), s. 615-618. ISSN 0362-4803. E-ISSN 1099-1344.
[International Isotope Symposium on the Synthesis and Applications of Isotopes and Isotopically Labelled Compounds /12./. Princeton, 07.06.2015-11.06.2015]
R&D Projects: GA MŠMT LG13002
Institutional support: RVO:61388963
Keywords : 6-amino-uracil derivatives * specific activity assay using NMR * [C-14]cyanoacetic acid
Subject RIV: CC - Organic Chemistry
Impact factor: 1.745, year: 2016
Permanent Link: http://hdl.handle.net/11104/0269008

7.

0476117 - ÚOCHB 2018 RIV NL eng J - Journal Article
Kolman, Viktor - Jansa, Petr - Kalčic, Filip - Janeba, Zlatko - Zídek, Zdeněk
Polysubstituted 4,6-bis(hetero)arylpyrimidines as dual inhibitors of nitric oxide and prostaglandin E-2 production.
Nitric Oxide-Biology and Chemistry. Roč. 67, Jul 1 (2017), s. 53-57. ISSN 1089-8603. E-ISSN 1089-8611
R&D Projects: GA TA ČR(CZ) TE01020028
Institutional support: RVO:61388963 ; RVO:68378041
Keywords : pyrimidine derivatives * nitric oxide * prostaglandin E-2 * dual inhibitors * anti-inflammatory properties
OECD category: Biochemistry and molecular biology; Organic chemistry (UEM-P)
Impact factor: 4.367, year: 2017
Permanent Link: http://hdl.handle.net/11104/0272652

8.

0493581 - ÚOCHB 2019 RIV FR eng J - Journal Article
Kolman, Viktor - Kalčic, Filip - Jansa, Petr - Zídek, Zdeněk - Janeba, Zlatko
Influence of the C-5 substitution in polysubstituted pyrimidines on inhibition of prostaglandin E2 production.
European Journal of Medicinal Chemistry. Roč. 156, Aug 5 (2018), s. 295-301. ISSN 0223-5234. E-ISSN 1768-3254
R&D Projects: GA TA ČR(CZ) TE01020028
Institutional support: RVO:61388963 ; RVO:68378041
Keywords : pyrimidines * Suzuki-Miyaura reaction * prostaglandin E2 * inhibitor
OECD category: Organic chemistry; Medicinal chemistry (UEM-P)
Impact factor: 4.833, year: 2018
Permanent Link: http://hdl.handle.net/11104/0286924

9.

0493604 - ÚOCHB 2019 RIV DE eng J - Journal Article
Česnek, Michal - Skácel, Jan - Jansa, Petr - Dračínský, Martin - Šmídková, Markéta - Mertlíková-Kaiserová, Helena - Soto-Velasquez, M. - Watts, V. J. - Janeba, Zlatko
Nucleobase Modified Adefovir (PMEA) Analogues as Potent and Selective Inhibitors of Adenylate Cyclases from Bordetella pertussis and Bacillus anthracis.
ChemMedChem. Roč. 13, č. 17 (2018), s. 1779-1796. ISSN 1860-7179. E-ISSN 1860-7187
R&D Projects: GA MV VG20102015046; GA ČR(CZ) GBP208/12/G016; GA MŠMT LO1302
Institutional support: RVO:61388963
Keywords : adefovir * adenylate cyclase * Bacillus anthracis * Bordetella pertussis * inhibitors
OECD category: Organic chemistry
Impact factor: 3.016, year: 2018
Permanent Link: http://hdl.handle.net/11104/0286939

10.

0500199 - ÚOCHB 2019 RIV GB eng J - Journal Article
Baszczyňski, Ondřej - Kaiser, Martin Maxmilian - Česnek, Michal - Břehová, Petra - Jansa, Petr - Procházková, Eliška - Dračínský, Martin - Snoeck, R. - Andrei, G. - Janeba, Zlatko
Xanthine-based acyclic nucleoside phosphonates with potent antiviral activity against varicella-zoster virus and human cytomegalovirus.
Antiviral Chemistry and Chemotherapy. Roč. 26, Nov 29 (2018), s. 1-13. ISSN 0956-3202
Institutional support: RVO:61388963
Keywords : acyclic nucleoside phosphonates * xanthine * PMEX * antiviral * HCMV * VZV
OECD category: Organic chemistry
https://journals.sagepub.com/doi/10.1177/2040206618813050
Permanent Link: http://hdl.handle.net/11104/0292843